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Save on Generic Levocetirizine 5 mg from India

The generic Xyzal 5 mg comes from India (Levorid) manufactured by Cipla. It is available in the quantity of 100 tablets.

Xyzal Information

Xyzal (levocetirizine) is a second-generation antihistamine used to relieve the symptoms of seasonal and perennial allergic rhinitis, such as sneezing, a runny and itchy nose, and watery eyes. It is also indicated for the treatment of chronic idiopathic urticaria (hives) and the associated itching. Levocetirizine is a metabolite of the popular second-generation antihistamine, cetirizine. It is the active enantiomer, or the pharmacologically active form, of cetirizine, meaning it is the part of the molecule that is responsible for the medication's effects. Because it is a purified form, it is highly potent, providing effective relief with a lower dose.

The mechanism of action for levocetirizine involves the selective blocking of the histamine H1 receptor. Histamine is a key chemical released by the body during an allergic reaction, and its interaction with H1 receptors is responsible for the classic symptoms of allergies. By blocking these receptors, Xyzal prevents histamine from triggering the allergic response, thereby reducing inflammation and symptoms. It has a very high affinity for the H1 receptor and a rapid onset of action, with effects often noticed within one hour. Because it is a second-generation antihistamine, it does not readily cross the blood-brain barrier at therapeutic doses, which is why it causes significantly less sedation than first-generation antihistamines like diphenhydramine.

In Canada, Xyzal is available over-the-counter in various formulations, including tablets and oral solutions. The standard dose for adults and children 12 years of age and older is 5 mg once daily, typically taken in the evening. For children aged 6 to 11, the dose is 2.5 mg once daily. Taking it in the evening is recommended due to the potential for mild drowsiness in some individuals. It provides 24-hour relief, making a once-daily dose convenient for most patients. It can be taken with or without food, as food does not significantly impact its absorption or effectiveness.

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Do I need a prescription to order Levocetirizine 5 mg ?

Yes, a prescription is required from your physician to order Levocetirizine 5 mg.